Detalles de la búsqueda
1.
New 1H-1,2,4-Triazolyl Derivatives as Antimicrobial Agents.
Chem Biodivers
; : e202400316, 2024 Feb 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-38422224
2.
In silico Design, Synthesis and Biological Evaluation of Novel Thieno[3,2-d]pyrimidine Derivatives for Cancer Therapy - A Preliminary Study on the Inhibitory Potential towards ATR Kinase Domain and PIKK Family.
Chem Biodivers
; 21(3): e202302071, 2024 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-38230843
3.
Substituted furan sulfonamides as carbonic anhydrase inhibitors: Synthesis, biological and in silico studies.
Bioorg Chem
; 138: 106621, 2023 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-37257407
4.
Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors.
Int J Mol Sci
; 24(3)2023 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-36769114
5.
Antimicrobial Activity of Some Steroidal Hydrazones.
Molecules
; 28(3)2023 Jan 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-36770834
6.
Discovery of Novel EGFR Inhibitor Targeting Wild-Type and Mutant Forms of EGFR: In Silico and In Vitro Study.
Molecules
; 28(7)2023 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-37049777
7.
New Bicyclic Pyridine-Based Hybrids Linked to the 1,2,3-Triazole Unit: Synthesis via Click Reaction and Evaluation of Neurotropic Activity and Molecular Docking.
Molecules
; 28(3)2023 Jan 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-36770592
8.
Identification of Novel Cyclooxygenase-1 Selective Inhibitors of Thiadiazole-Based Scaffold as Potent Anti-Inflammatory Agents with Safety Gastric and Cytotoxic Profile.
Molecules
; 28(8)2023 Apr 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-37110650
9.
Developing New Treatments for COVID-19 through Dual-Action Antiviral/Anti-Inflammatory Small Molecules and Physiologically Based Pharmacokinetic Modeling.
Int J Mol Sci
; 23(14)2022 07 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-35887353
10.
Enhancement of the Anti-Inflammatory Activity of NSAIDs by Their Conjugation with 3,4,5-Trimethoxybenzyl Alcohol.
Molecules
; 27(7)2022 Mar 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-35408503
11.
Benzothiazole and Chromone Derivatives as Potential ATR Kinase Inhibitors and Anticancer Agents.
Molecules
; 27(14)2022 Jul 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-35889508
12.
Thiazolidin-4-Ones as Potential Antimicrobial Agents: Experimental and In Silico Evaluation.
Molecules
; 27(6)2022 Mar 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-35335296
13.
Thiazole/Thiadiazole/Benzothiazole Based Thiazolidin-4-One Derivatives as Potential Inhibitors of Main Protease of SARS-CoV-2.
Molecules
; 27(7)2022 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-35408577
14.
Discovery of 5-Methylthiazole-Thiazolidinone Conjugates as Potential Anti-Inflammatory Agents: Molecular Target Identification and In Silico Studies.
Molecules
; 27(23)2022 Nov 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-36500230
15.
Synthesis, Biological Evaluation and Molecular Docking Studies of 5-Indolylmethylen-4-oxo-2-thioxothiazolidine Derivatives.
Molecules
; 27(3)2022 Feb 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35164333
16.
2-Aryl-3-(6-trifluoromethoxy)benzo[d]thiazole-based thiazolidinone hybrids as potential anti-infective agents: Synthesis, biological evaluation and molecular docking studies.
Bioorg Med Chem Lett
; 32: 127718, 2021 01 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-33253880
17.
Synthesis and antimicrobial activity of new 2-piperazin-1-yl-N-1,3-thiazol-2-ylacetamides of cyclopenta[c]pyridines and pyrano[3,4-c]pyridines.
Arch Pharm (Weinheim)
; 354(1): e2000208, 2021 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-33029832
18.
Chromene-Containing Aromatic Sulfonamides with Carbonic Anhydrase Inhibitory Properties.
Int J Mol Sci
; 22(10)2021 May 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-34064890
19.
Thiazole Ring-A Biologically Active Scaffold.
Molecules
; 26(11)2021 May 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-34070661
20.
Carbonic Anhydrase Inhibition with Sulfonamides Incorporating Pyrazole- and Pyridazinecarboxamide Moieties Provides Examples of Isoform-Selective Inhibitors.
Molecules
; 26(22)2021 Nov 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-34834114